| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Translocator protein |
|---|
| Ligand | BDBM98175 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | In Vitro Binding Assay |
|---|
| Ki | 10.96±0.0 nM |
|---|
| Citation |  Kassiou, M; James, ML; Luus, CA Translocator protein ligands US Patent US8492379 Publication Date 7/23/2013 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Translocator protein |
|---|
| Name: | Translocator protein |
|---|
| Synonyms: | BZRP | MBR | Mitochondrial benzodiazepine receptor | PBR | PKBS | Peripheral benzodiazepine receptor-related protein | Peripheral-type benzodiazepine receptor | TSPO | TSPO_HUMAN |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 18834.74 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P30536 |
|---|
| Residue: | 169 |
|---|
| Sequence: | MAPPWVPAMGFTLAPSLGCFVGSRFVHGEGLRWYAGLQKPSWHPPHWVLGPVWGTLYSAM
GYGSYLVWKELGGFTEKAVVPLGLYTGQLALNWAWPPIFFGARQMGWALVDLLLVSGAAA
ATTVAWYQVSPLAARLLYPYLAWLAFTTTLNYCVWRDNHGWRGGRRLPE
|
|
|
|---|
| BDBM98175 |
|---|
| n/a |
|---|
| Name | BDBM98175 |
|---|
| Synonyms: | US8492379, 52 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C20H24N4O2 |
|---|
| Mol. Mass. | 352.4302 |
|---|
| SMILES | CCN(CC)C(=O)Cc1c(nc2c(C)cc(C)nn12)-c1ccc(O)cc1 |
|---|
| Structure | 
|
|---|
Search and Browse
