| Reaction Details |
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 | Report a problem with these data |
| Target | Reverse transcriptase protein |
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| Ligand | BDBM2161 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Enzyme Inhibition Assay |
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| IC50 | 21760±n/a nM |
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| Citation |  Bode, ML; Rousseau, AL; Gravestock, D; Moleele, SS; Van Der Westhuyzen, CW Imidazopyridines and imidazopyrimidines as HIV-1 reverse transcriptase inhibitors US Patent US8501767 Publication Date 8/6/2013 |
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| More Info.: | Get all data from this article, Assay Method |
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| Reverse transcriptase protein |
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| Name: | Reverse transcriptase protein |
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| Synonyms: | n/a |
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| Type: | Protein |
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| Mol. Mass.: | 30157.99 |
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| Organism: | Human immunodeficiency virus 1 |
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| Description: | Q9WJP9 |
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| Residue: | 259 |
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| Sequence: | PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTELEKEGKNSKIGPENPYNTPV
FAIKKKDSTKWRKLVDFRELNRKTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPL
DKDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVI
YQYMDDLYVGSDLEIGQHRTKIEELRQHLLKWGFYTPDKKHQKEPPFLWMGYELHPDKWT
VQPIVLPEKDSWTVNDIQK
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| BDBM2161 |
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| n/a |
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| Name | BDBM2161 |
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| Synonyms: | DG 402-49686 | US8501787, 89 |
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| Type | n/a |
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| Emp. Form. | C19H19Cl2N3 |
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| Mol. Mass. | 360.28 |
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| SMILES | Clc1ccc(-c2nc3ccccn3c2NC2CCCCC2)c(Cl)c1 |
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| Structure | 
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