| Reaction Details |
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 | Report a problem with these data |
| Target | Kallikrein-7 |
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| Ligand | BDBM51528 |
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| Substrate/Competitor | n/a |
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| EC50 | 3623±n/a nM |
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| Citation |  PubChem, PC Fluorescence Intensity-based biochemical primary high throughput dose response assay to identify activators of kallikrein-7 (K7) zymogen PubChem Bioassay(2013)[AID] |
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| More Info.: | Get all data from this article |
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| Kallikrein-7 |
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| Name: | Kallikrein-7 |
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| Synonyms: | KLK7 | KLK7_HUMAN | Kallikrein 7 | Kallikrein-7 | PRSS6 | SCCE | Serine protease 6 | Stratum corneum chymotryptic enzyme | hK7 | hSCCE | kallikrein-7 isoform 1 preproprotein |
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| Type: | PROTEIN |
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| Mol. Mass.: | 27535.05 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1469257 |
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| Residue: | 253 |
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| Sequence: | MARSLLLPLQILLLSLALETAGEEAQGDKIIDGAPCARGSHPWQVALLSGNQLHCGGVLV
NERWVLTAAHCKMNEYTVHLGSDTLGDRRAQRIKASKSFRHPGYSTQTHVNDLMLVKLNS
QARLSSMVKKVRLPSRCEPPGTTCTVSGWGTTTSPDVTFPSDLMCVDVKLISPQDCTKVY
KDLLENSMLCAGIPDSKKNACNGDSGGPLVCRGTLQGLVSWGTFPCGQPNDPGVYTQVCK
FTKWINDTMKKHR
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| BDBM51528 |
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| n/a |
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| Name | BDBM51528 |
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| Synonyms: | 2-amino-1-(2-piperidinoethyl)pyrrolo[3,2-b]quinoxaline-3-carboxylic acid ethyl ester | 2-amino-1-[2-(1-piperidinyl)ethyl]-3-pyrrolo[3,2-b]quinoxalinecarboxylic acid ethyl ester | MLS000056772 | SMR000065736 | cid_1888166 | ethyl 2-amino-1-(2-piperidin-1-ylethyl)pyrrolo[3,2-b]quinoxaline-3-carboxylate | ethyl 2-azanyl-1-(2-piperidin-1-ylethyl)pyrrolo[3,2-b]quinoxaline-3-carboxylate |
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| Type | Small organic molecule |
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| Emp. Form. | C20H25N5O2 |
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| Mol. Mass. | 367.4448 |
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| SMILES | CCOC(=O)c1c(N)n(CCN2CCCCC2)c2nc3ccccc3nc12 |
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| Structure | 
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