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TargetKallikrein-7
LigandBDBM100118
Substrate/Competitorn/a
EC50 5160±n/a nM
Citation PubChem, PC Fluorescence Intensity-based biochemical primary high throughput dose response assay to identify activators of kallikrein-7 (K7) zymogen PubChem Bioassay(2013)[AID]
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Kallikrein-7
Name:Kallikrein-7
Synonyms:KLK7 | KLK7_HUMAN | Kallikrein 7 | Kallikrein-7 | PRSS6 | SCCE | Serine protease 6 | Stratum corneum chymotryptic enzyme | hK7 | hSCCE | kallikrein-7 isoform 1 preproprotein
Type:PROTEIN
Mol. Mass.:27535.05
Organism:Homo sapiens (Human)
Description:ChEMBL_1469257
Residue:253
Sequence:
MARSLLLPLQILLLSLALETAGEEAQGDKIIDGAPCARGSHPWQVALLSGNQLHCGGVLV
NERWVLTAAHCKMNEYTVHLGSDTLGDRRAQRIKASKSFRHPGYSTQTHVNDLMLVKLNS
QARLSSMVKKVRLPSRCEPPGTTCTVSGWGTTTSPDVTFPSDLMCVDVKLISPQDCTKVY
KDLLENSMLCAGIPDSKKNACNGDSGGPLVCRGTLQGLVSWGTFPCGQPNDPGVYTQVCK
FTKWINDTMKKHR
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BDBM100118
n/a
NameBDBM100118
Synonyms:2-(2-keto-3-phenyl-chromen-7-yl)oxypropionic acid methyl ester | 2-[(2-oxo-3-phenyl-1-benzopyran-7-yl)oxy]propanoic acid methyl ester | MLS001167026 | SMR000641318 | cid_16450243 | methyl 2-(2-oxidanylidene-3-phenyl-chromen-7-yl)oxypropanoate | methyl 2-(2-oxo-3-phenylchromen-7-yl)oxypropanoate
TypeSmall organic molecule
Emp. Form.C19H16O5
Mol. Mass.324.3273
SMILESCOC(=O)C(C)Oc1ccc2cc(-c3ccccc3)c(=O)oc2c1
Structure
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