| Reaction Details |
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 | Report a problem with these data |
| Target | COUP transcription factor 2 |
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| Ligand | BDBM75744 |
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| Substrate/Competitor | n/a |
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| IC50 | 2750±n/a nM |
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| Citation |  PubChem, PC Luminescence-based cell-based high throughput dose response assay to identify inhibitors of COUP-TFII (NR2F2) PubChem Bioassay(2013)[AID] |
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| More Info.: | Get all data from this article |
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| COUP transcription factor 2 |
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| Name: | COUP transcription factor 2 |
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| Synonyms: | ARP1 | COT2_HUMAN | COUP transcription factor 2 isoform a | NR2F2 | TFCOUP2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 45583.83 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_14149746 |
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| Residue: | 414 |
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| Sequence: | MAMVVSTWRDPQDEVPGSQGSQASQAPPVPGPPPGAPHTPQTPGQGGPASTPAQTAAGGQ
GGPGGPGSDKQQQQQHIECVVCGDKSSGKHYGQFTCEGCKSFFKRSVRRNLSYTCRANRN
CPIDQHHRNQCQYCRLKKCLKVGMRREAVQRGRMPPTQPTHGQFALTNGDPLNCHSYLSG
YISLLLRAEPYPTSRFGSQCMQPNNIMGIENICELAARMLFSAVEWARNIPFFPDLQITD
QVALLRLTWSELFVLNAAQCSMPLHVAPLLAAAGLHASPMSADRVVAFMDHIRIFQEQVE
KLKALHVDSAEYSCLKAIVLFTSDACGLSDVAHVESLQEKSQCALEEYVRSQYPNQPTRF
GKLLLRLPSLRTVSSSVIEQLFFVRLVGKTPIETLIRDMLLSGSSFNWPYMAIQ
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| BDBM75744 |
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| n/a |
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| Name | BDBM75744 |
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| Synonyms: | (2E)-3-ethyl-2-[(1-ethyl-2-quinolin-1-iumyl)methylidene]-6-methyl-1,3-benzothiazole;iodide | (2E)-3-ethyl-2-[(1-ethylquinolin-1-ium-2-yl)methylene]-6-methyl-1,3-benzothiazole;iodide | (2E)-3-ethyl-2-[(1-ethylquinolin-1-ium-2-yl)methylidene]-6-methyl-1,3-benzothiazole;iodide | MLS000688479 | SMR000284410 | cid_16187754 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H23N2S |
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| Mol. Mass. | 347.496 |
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| SMILES | CCN1\C(Sc2cc(C)ccc12)=C/c1ccc2ccccc2[n+]1CC |
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| Structure | 
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