| Reaction Details |
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 | Report a problem with these data |
| Target | Transcription initiation factor IIA subunit 1 |
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| Ligand | BDBM108117 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Inhibition Assay |
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| Ki | 1200±0.0 nM |
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| Citation |  Herold, P; Daghish, M; Jelakovic, S; Ludwig, F; Reichelt, C; Schulze, A; Schweinitz, A Trypsin-like serine protease inhibitors, and their preparation and use US Patent US8598206 Publication Date 12/3/2013 |
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| More Info.: | Get all data from this article, Assay Method |
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| Transcription initiation factor IIA subunit 1 |
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| Name: | Transcription initiation factor IIA subunit 1 |
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| Synonyms: | GTF2A1 | TF2A1 | TF2AA_HUMAN | Transcription initiation factor IIA |
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| Type: | Enzyme |
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| Mol. Mass.: | 41485.12 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P52655 |
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| Residue: | 376 |
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| Sequence: | MANSANTNTVPKLYRSVIEDVINDVRDIFLDDGVDEQVLMELKTLWENKLMQSRAVDGFH
SEEQQLLLQVQQQHQPQQQQHHHHHHHQQAQPQQTVPQQAQTQQVLIPASQQATAPQVIV
PDSKLIQHMNASNMSAAATAATLALPAGVTPVQQILTNSGQLLQVVRAANGAQYIFQPQQ
SVVLQQQVIPQMQPGGVQAPVIQQVLAPLPGGISPQTGVIIQPQQILFTGNKTQVIPTTV
AAPTPAQAQITATGQQQPQAQPAQTQAPLVLQVDGTGDTSSEEDEDEEEDYDDDEEEDKE
KDGAEDGQVEEEPLNSEDDVSDEEGQELFDTENVVVCQYDKIHRSKNKWKFHLKDGIMNL
NGRDYIFSKAIGDAEW
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| BDBM108117 |
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| n/a |
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| Name | BDBM108117 |
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| Synonyms: | US8598206, Table 6, 2 |
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| Type | Small organic molecule |
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| Emp. Form. | C34H45N7O4S |
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| Mol. Mass. | 647.831 |
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| SMILES | NC(=N)c1ccc(CNC(=O)[C@H](CCC2CCNCC2)NC(=O)[C@@H](CCCc2ccncc2)NS(=O)(=O)Cc2ccccc2)cc1 |r| |
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| Structure | 
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