Reaction Details |
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Target | Transcription initiation factor IIA subunit 1 |
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Ligand | BDBM47177 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Inhibition Assay |
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Ki | 3800±0.0 nM |
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Citation | Herold, P; Daghish, M; Jelakovic, S; Ludwig, F; Reichelt, C; Schulze, A; Schweinitz, A Trypsin-like serine protease inhibitors, and their preparation and use US Patent US8598206 Publication Date 12/3/2013 |
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More Info.: | Get all data from this article, Assay Method |
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Transcription initiation factor IIA subunit 1 |
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Name: | Transcription initiation factor IIA subunit 1 |
Synonyms: | GTF2A1 | TF2A1 | TF2AA_HUMAN | Transcription initiation factor IIA |
Type: | Enzyme |
Mol. Mass.: | 41485.12 |
Organism: | Homo sapiens (Human) |
Description: | P52655 |
Residue: | 376 |
Sequence: | MANSANTNTVPKLYRSVIEDVINDVRDIFLDDGVDEQVLMELKTLWENKLMQSRAVDGFH
SEEQQLLLQVQQQHQPQQQQHHHHHHHQQAQPQQTVPQQAQTQQVLIPASQQATAPQVIV
PDSKLIQHMNASNMSAAATAATLALPAGVTPVQQILTNSGQLLQVVRAANGAQYIFQPQQ
SVVLQQQVIPQMQPGGVQAPVIQQVLAPLPGGISPQTGVIIQPQQILFTGNKTQVIPTTV
AAPTPAQAQITATGQQQPQAQPAQTQAPLVLQVDGTGDTSSEEDEDEEEDYDDDEEEDKE
KDGAEDGQVEEEPLNSEDDVSDEEGQELFDTENVVVCQYDKIHRSKNKWKFHLKDGIMNL
NGRDYIFSKAIGDAEW
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BDBM47177 |
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n/a |
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Name | BDBM47177 |
Synonyms: | BDBM108100 | US8598206, Table 6, 9 |
Type | n/a |
Emp. Form. | C36H53N7O5S |
Mol. Mass. | 695.915 |
SMILES | CC(=O)N1CCC(CCC[C@@H](NS(=O)(=O)Cc2ccccc2)C(=O)N[C@@H](CCC2CCNCC2)C(=O)NCc2ccc(cc2)C(N)=N)CC1 |r| |
Structure |
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