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TargetTranscription initiation factor IIA
LigandBDBM108102
Substrate/Competitorn/a
Meas. Tech.Inhibition Assay
Ki 4500±0.0 nM
Citation Herold PDaghish MJelakovic SLudwig FReichelt CSchulze ASchweinitz A Trypsin-like serine protease inhibitors, and their preparation and use US Patent  US8598206 Publication Date 12/3/2013
More Info.:Get all data from this article,  Assay Method
 
Transcription initiation factor IIA
Name:Transcription initiation factor IIA
Synonyms:n/a
Type:Enzyme
Mol. Mass.:41485.12
Organism:Homo sapiens (Human)
Description:P52655
Residue:376
Sequence:
MANSANTNTVPKLYRSVIEDVINDVRDIFLDDGVDEQVLMELKTLWENKLMQSRAVDGFH
SEEQQLLLQVQQQHQPQQQQHHHHHHHQQAQPQQTVPQQAQTQQVLIPASQQATAPQVIV
PDSKLIQHMNASNMSAAATAATLALPAGVTPVQQILTNSGQLLQVVRAANGAQYIFQPQQ
SVVLQQQVIPQMQPGGVQAPVIQQVLAPLPGGISPQTGVIIQPQQILFTGNKTQVIPTTV
AAPTPAQAQITATGQQQPQAQPAQTQAPLVLQVDGTGDTSSEEDEDEEEDYDDDEEEDKE
KDGAEDGQVEEEPLNSEDDVSDEEGQELFDTENVVVCQYDKIHRSKNKWKFHLKDGIMNL
NGRDYIFSKAIGDAEW
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  Blast E-value cutoff:
BDBM108102
n/a
NameBDBM108102
Synonyms:US8598206, Table 6, 11
TypeSmall organic molecule
Emp. Form.C36H53N7O6S
Mol. Mass.711.914
SMILESCOCC(=O)N1CCC(CC[C@@H](NS(=O)(=O)Cc2ccccc2)C(=O)N[C@@H](CCC2CCNCC2)C(=O)NCc2ccc(cc2)C(N)=N)CC1 |r|
Structure
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