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TargetHistone H1.0
LigandBDBM50130293
Substrate/Competitorn/a
Meas. Tech.Binding Assay
Ki 28±0.0 nM
Citation Mates, SFienberg, AWennogle, L Methods and compositions for sleep disorders and other disorders US Patent US8598119 Publication Date 12/3/2013
More Info.:Get all data from this article,  Assay Method
 
Histone H1.0
Name:Histone H1.0
Synonyms:H1-0 | H10_HUMAN | H1F0 | H1FV | Histone H1
Type:Cell-surface receptors
Mol. Mass.:20917.09
Organism:Homo sapiens (Human)
Description:P07305
Residue:194
Sequence:
MTENSTSAPAAKPKRAKASKKSTDHPKYSDMIVAAIQAEKNRAGSSRQSIQKYIKSHYKV
GENADSQIKLSIKRLVTTGVLKQTKGVGASGSFRLAKSDEPKKSVAFKKTKKEIKKVATP
KKASKPKKAASKAPTKKPKATPVKKAKKKLAATPKKAKKPKTVKAKPVKASKPKKAKPVK
PKAKSSAKRAGKKK
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50130293
n/a
NameBDBM50130293
Synonyms:7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}-3,4-dihydroquinolin-2(1H)-one | ARIPIPRAZOLE | CHEMBL1112 | US10174011, aripiprazole | US10752588, Compound Aripiprazole | US11498896, Compound Aripiprazole | US9018213, aripprazole | US9156822, Aripiprazole
TypeSmall organic molecule
Emp. Form.C23H27Cl2N3O2
Mol. Mass.448.385
SMILESClc1cccc(N2CCN(CCCCOc3ccc4CCC(=O)Nc4c3)CC2)c1Cl
Structure
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