| Reaction Details |
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 | Report a problem with these data |
| Target | Stromelysin-2 |
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| Ligand | BDBM120159 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Inhibition Assay |
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| Ki | 111±n/a nM |
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| Citation |  Devel, L; Beau, F; Czarny, B; Dive, V Pseudodipeptides as MMP inhibitors US Patent US8691753 Publication Date 4/8/2014 |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Stromelysin-2 |
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| Name: | Stromelysin-2 |
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| Synonyms: | MMP10 | MMP10_HUMAN | Matrix Metalloproteinase-10 (MMP-10) | Matrix metalloproteinase 10 | STMY2 |
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| Type: | Enzyme |
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| Mol. Mass.: | 54143.02 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P09238 |
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| Residue: | 476 |
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| Sequence: | MMHLAFLVLLCLPVCSAYPLSGAAKEEDSNKDLAQQYLEKYYNLEKDVKQFRRKDSNLIV
KKIQGMQKFLGLEVTGKLDTDTLEVMRKPRCGVPDVGHFSSFPGMPKWRKTHLTYRIVNY
TPDLPRDAVDSAIEKALKVWEEVTPLTFSRLYEGEADIMISFAVKEHGDFYSFDGPGHSL
AHAYPPGPGLYGDIHFDDDEKWTEDASGTNLFLVAAHELGHSLGLFHSANTEALMYPLYN
SFTELAQFRLSQDDVNGIQSLYGPPPASTEEPLVPTKSVPSGSEMPAKCDPALSFDAIST
LRGEYLFFKDRYFWRRSHWNPEPEFHLISAFWPSLPSYLDAAYEVNSRDTVFIFKGNEFW
AIRGNEVQAGYPRGIHTLGFPPTIRKIDAAVSDKEKKKTYFFAADKYWRFDENSQSMEQG
FPRLIADDFPGVEPKVDAVLQAFGFFYFFSGSSQFEFDPNARMVTHILKSNSWLHC
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| BDBM120159 |
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| n/a |
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| Name | BDBM120159 |
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| Synonyms: | US8691753, 7 |
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| Type | Small organic molecule |
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| Emp. Form. | C28H29ClN4O8 |
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| Mol. Mass. | 585.005 |
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| SMILES | NC(=O)[C@@H](CCC(O)=O)NC(=O)[C@@H](CCC(O)=O)NC(=O)CCc1cc(no1)-c1ccc(cc1)-c1cccc(Cl)c1 |r| |
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| Structure | 
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