| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Stromelysin-2 |
|---|
| Ligand | BDBM120219 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Inhibition Assay |
|---|
| Ki | 71±n/a nM |
|---|
| Citation |  Devel, L; Beau, F; Czarny, B; Dive, V Pseudodipeptides as MMP inhibitors US Patent US8691753 Publication Date 4/8/2014 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Stromelysin-2 |
|---|
| Name: | Stromelysin-2 |
|---|
| Synonyms: | MMP10 | MMP10_HUMAN | Matrix Metalloproteinase-10 (MMP-10) | Matrix metalloproteinase 10 | STMY2 |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 54143.02 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P09238 |
|---|
| Residue: | 476 |
|---|
| Sequence: | MMHLAFLVLLCLPVCSAYPLSGAAKEEDSNKDLAQQYLEKYYNLEKDVKQFRRKDSNLIV
KKIQGMQKFLGLEVTGKLDTDTLEVMRKPRCGVPDVGHFSSFPGMPKWRKTHLTYRIVNY
TPDLPRDAVDSAIEKALKVWEEVTPLTFSRLYEGEADIMISFAVKEHGDFYSFDGPGHSL
AHAYPPGPGLYGDIHFDDDEKWTEDASGTNLFLVAAHELGHSLGLFHSANTEALMYPLYN
SFTELAQFRLSQDDVNGIQSLYGPPPASTEEPLVPTKSVPSGSEMPAKCDPALSFDAIST
LRGEYLFFKDRYFWRRSHWNPEPEFHLISAFWPSLPSYLDAAYEVNSRDTVFIFKGNEFW
AIRGNEVQAGYPRGIHTLGFPPTIRKIDAAVSDKEKKKTYFFAADKYWRFDENSQSMEQG
FPRLIADDFPGVEPKVDAVLQAFGFFYFFSGSSQFEFDPNARMVTHILKSNSWLHC
|
|
|
|---|
| BDBM120219 |
|---|
| n/a |
|---|
| Name | BDBM120219 |
|---|
| Synonyms: | US8691753, 68 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C29H31N3O6 |
|---|
| Mol. Mass. | 517.5729 |
|---|
| SMILES | NC(=O)[C@H](CO)NC(=O)[C@H](CCC(O)=O)NC(=O)CCc1ccc(cc1)-c1ccc(cc1)-c1ccccc1 |r| |
|---|
| Structure | 
|
|---|
Search and Browse
