| Reaction Details |
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 | Report a problem with these data |
| Target | Prokineticin receptor 2 |
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| Ligand | BDBM121070 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Calcium Mobilization Assay |
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| Temperature | 310.15±n/a K |
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| Ki | 0.81±n/a nM |
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| Comments | extracted |
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| Citation |  Zhou, Q; Li, J; Huang, Q Prokineticin receptor antagonists and uses thereof US Patent US8722896 Publication Date 5/13/2014 |
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| More Info.: | Get all data from this article, Assay Method |
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| Prokineticin receptor 2 |
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| Name: | Prokineticin receptor 2 |
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| Synonyms: | Prokineticin receptor 2 (PRK2) |
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| Type: | Enzyme |
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| Mol. Mass.: | 44473.96 |
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| Organism: | Cricetulus griseus (Chinese hamster) |
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| Description: | G3H407 |
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| Residue: | 391 |
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| Sequence: | MPPAGINMASQNKNTSFAPDLNPSQDHISSLPFNFSYSDYDLPLDGDEDMTKTQTFFAAK
IVIGVALAGIMLVCGIGNFVFIAALARYKKLRNLTNLLIANLAISDFLVAIVCCPFEMDY
YVVRQLSWEHGHVLCASVNYLRTVSLYVSTNALLAIAIDRYLAIVHPLKPRMNYQTASFL
IALVWMVSILIAIPSAYFTTETILDIVKNQEKIFCGQIWPVDQQLYYKSYFLFVFGLEFV
GPVVAMTLCYARISQELWFKAVPGFQTEQIRKRLRCRRKTVLLLMGILTAYVLCWAPFYG
FTIVRDFFPTVFVKEKHYLTAFYVVECIAMSNSMINTICFVTVKNNTMKYFKKMLLLHWQ
PSRYGSKSSADLDLKTSGVPATEEVDCIRLK
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| BDBM121070 |
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| n/a |
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| Name | BDBM121070 |
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| Synonyms: | US8722896, (-)-(3R)-1-(2-Methoxybenzyl)- N-(9-fluoro-3,4-dihydro-2H-1,5- benzodioxepin-7-ylmethyl)-N- isobutylpyrrolidine-3- carboxamide |
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| Type | Small organic molecule |
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| Emp. Form. | C27H35FN2O4 |
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| Mol. Mass. | 470.5762 |
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| SMILES | COc1ccccc1CN1CC[C@H](C1)C(=O)N(CC(C)C)Cc1cc(F)c2OCCCOc2c1 |r| |
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| Structure | 
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