Reaction Details |
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Target | Somatostatin receptor type 5 |
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Ligand | BDBM123236 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Binding Assay |
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pH | 7.8±n/a |
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IC50 | 0.4374±n/a nM |
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Comments | extracted |
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Citation | Duffy, JL; Bao, J; Ondeyka, DL; Tyagarajan, S; Shao, P; Ye, F; Katipally, R; Zwicker, A; Sherer, EC; Plotkin, MA; Moningka, R; Hussain, Z; Wood, HB; Ujjainwalla, F; Romero, FA; Finke, PE; Zang, Y; Liu, W Spiroxazolidinone compounds US Patent US8742110 Publication Date 6/3/2014 |
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More Info.: | Get all data from this article, Assay Method |
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Somatostatin receptor type 5 |
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Name: | Somatostatin receptor type 5 |
Synonyms: | SOMATOSTATIN SST5 | SS-5-R | SS5-R | SS5R | SSR5_HUMAN | SSTR5 | Somatostatin receptor type 5 (SSTR5) |
Type: | Enzyme |
Mol. Mass.: | 39218.02 |
Organism: | Homo sapiens (Human) |
Description: | P35346 |
Residue: | 364 |
Sequence: | MEPLFPASTPSWNASSPGAASGGGDNRTLVGPAPSAGARAVLVPVLYLLVCAAGLGGNTL
VIYVVLRFAKMKTVTNIYILNLAVADVLYMLGLPFLATQNAASFWPFGPVLCRLVMTLDG
VNQFTSVFCLTVMSVDRYLAVVHPLSSARWRRPRVAKLASAAAWVLSLCMSLPLLVFADV
QEGGTCNASWPEPVGLWGAVFIIYTAVLGFFAPLLVICLCYLLIVVKVRAAGVRVGCVRR
RSERKVTRMVLVVVLVFAGCWLPFFTVNIVNLAVALPQEPASAGLYFFVVILSYANSCAN
PVLYGFLSDNFRQSFQKVLCLRKGSGAKDADATEPRPDRIRQQQEATPPAHRAAANGLMQ
TSKL
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BDBM123236 |
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n/a |
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Name | BDBM123236 |
Synonyms: | US8742110, 3-21 |
Type | Small organic molecule |
Emp. Form. | C31H32F2N2O6 |
Mol. Mass. | 566.5924 |
SMILES | CCOc1cc(CN2CCC3(CN(C(=O)O3)c3ccc(cc3F)C(O)=O)CC2)cc(OCC)c1-c1ccc(F)cc1 |
Structure |
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