| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Somatostatin receptor type 5 |
|---|
| Ligand | BDBM123307 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Binding Assay |
|---|
| pH | 7.8±n/a |
|---|
| IC50 | 0.5502±n/a nM |
|---|
| Comments | extracted |
|---|
| Citation |  Duffy, JL; Bao, J; Ondeyka, DL; Tyagarajan, S; Shao, P; Ye, F; Katipally, R; Zwicker, A; Sherer, EC; Plotkin, MA; Moningka, R; Hussain, Z; Wood, HB; Ujjainwalla, F; Romero, FA; Finke, PE; Zang, Y; Liu, W Spiroxazolidinone compounds US Patent US8742110 Publication Date 6/3/2014 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Somatostatin receptor type 5 |
|---|
| Name: | Somatostatin receptor type 5 |
|---|
| Synonyms: | SOMATOSTATIN SST5 | SS-5-R | SS5-R | SS5R | SSR5_HUMAN | SSTR5 | Somatostatin receptor type 5 (SSTR5) |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 39218.02 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P35346 |
|---|
| Residue: | 364 |
|---|
| Sequence: | MEPLFPASTPSWNASSPGAASGGGDNRTLVGPAPSAGARAVLVPVLYLLVCAAGLGGNTL
VIYVVLRFAKMKTVTNIYILNLAVADVLYMLGLPFLATQNAASFWPFGPVLCRLVMTLDG
VNQFTSVFCLTVMSVDRYLAVVHPLSSARWRRPRVAKLASAAAWVLSLCMSLPLLVFADV
QEGGTCNASWPEPVGLWGAVFIIYTAVLGFFAPLLVICLCYLLIVVKVRAAGVRVGCVRR
RSERKVTRMVLVVVLVFAGCWLPFFTVNIVNLAVALPQEPASAGLYFFVVILSYANSCAN
PVLYGFLSDNFRQSFQKVLCLRKGSGAKDADATEPRPDRIRQQQEATPPAHRAAANGLMQ
TSKL
|
|
|
|---|
| BDBM123307 |
|---|
| n/a |
|---|
| Name | BDBM123307 |
|---|
| Synonyms: | US8742110, 6-25 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C26H28BrN3O4 |
|---|
| Mol. Mass. | 526.422 |
|---|
| SMILES | CC(C)n1cc(CN2CCC3(CN(C(=O)O3)c3ccc(cc3)C(O)=O)CC2)c2cc(Br)ccc12 |
|---|
| Structure | 
|
|---|
Search and Browse
