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TargetCore-binding factor subunit beta
LigandBDBM123676
Substrate/Competitorn/a
Meas. Tech.FRET Assay
IC50 3400±n/a nM
Citation Bushweller, JHGrembecka, JIllendula, ADixon, L Inhibitors of inv(16) leukemia US Patent US8748618 Publication Date 6/10/2014
More Info.:Get all data from this article,  Assay Method
 
Core-binding factor subunit beta
Name:Core-binding factor subunit beta
Synonyms:CBFB | Core-binding factor subunit beta (CBFB) | PEBB_HUMAN
Type:Enzyme
Mol. Mass.:21507.90
Organism:Homo sapiens (Human)
Description:Q13951
Residue:182
Sequence:
MPRVVPDQRSKFENEEFFRKLSRECEIKYTGFRDRPHEERQARFQNACRDGRSEIAFVAT
GTNLSLQFFPASWQGEQRQTPSREYVDLEREAGKVYLKAPMILNGVCVIWKGWIDLQRLD
GMGCLEFDEERAQQEDALAQQAFEEARRRTREFEDRDRSHREEMEVRVSQLLAVTGKKTT
RP
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BDBM123676
n/a
NameBDBM123676
Synonyms:US8748618, AI-10-88
TypeSmall organic molecule
Emp. Form.C15H11N5
Mol. Mass.261.2813
SMILESc1cn(cn1)-c1ccc2[nH]c(nc2c1)-c1ccccn1
Structure
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