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TargetIntegrin-linked protein kinase
LigandBDBM123936
Substrate/Competitorn/a
Meas. Tech.In Vitro Ezyme Assay
Temperature313.15±n/a K
IC50 70±n/a nM
Commentsextracted
Citation Zhang, ZDaynard, TSWang, SDu, XChopiuk, GBYan, JChen, JSviridov, SV Pyrazolylbenzothiazole derivatives and their use as therapeutic agents US Patent US8754233 Publication Date 6/17/2014
More Info.:Get all data from this article,  Assay Method
 
Integrin-linked protein kinase
Name:Integrin-linked protein kinase
Synonyms:ILK | ILK1 | ILK2 | ILK_HUMAN | Integrin-linked protein kinase (ILK) | Serine/threonine-protein kinase ILK-1
Type:Protein
Mol. Mass.:51429.75
Organism:Homo sapiens (Human)
Description:Q13418
Residue:452
Sequence:
MDDIFTQCREGNAVAVRLWLDNTENDLNQGDDHGFSPLHWACREGRSAVVEMLIMRGARI
NVMNRGDDTPLHLAASHGHRDIVQKLLQYKADINAVNEHGNVPLHYACFWGQDQVAEDLV
ANGALVSICNKYGEMPVDKAKAPLRELLRERAEKMGQNLNRIPYKDTFWKGTTRTRPRNG
TLNKHSGIDFKQLNFLTKLNENHSGELWKGRWQGNDIVVKVLKVRDWSTRKSRDFNEECP
RLRIFSHPNVLPVLGACQSPPAPHPTLITHWMPYGSLYNVLHEGTNFVVDQSQAVKFALD
MARGMAFLHTLEPLIPRHALNSRSVMIDEDMTARISMADVKFSFQCPGRMYAPAWVAPEA
LQKKPEDTNRRSADMWSFAVLLWELVTREVPFADLSNMEIGMKVALEGLRPTIPPGISPH
VCKLMKICMNEDPAKRPKFDMIVPILEKMQDK
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  Blast E-value cutoff:
BDBM123936
n/a
NameBDBM123936
Synonyms:US8754233, 2-(3-Amino-5-methyl-1H-pyrazol-4-yl)-benzothiazole-6-sulfonic acid methyl amide
TypeSmall organic molecule
Emp. Form.C12H13N5O2S2
Mol. Mass.323.394
SMILESCNS(=O)(=O)c1ccc2nc(sc2c1)-c1c(C)[nH]nc1N
Structure
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