| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Calcitonin gene-related peptide 1 |
|---|
| Ligand | BDBM126180 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Binding Assay |
|---|
| pH | 7.4±n/a |
|---|
| Temperature | 298.15±n/a K |
|---|
| Ki | 58±n/a nM |
|---|
| Comments | extracted |
|---|
| Citation |  Stump, CA; Quigley, AG CGRP receptor antagonists US Patent US8778957 Publication Date 7/15/2014 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Calcitonin gene-related peptide 1 |
|---|
| Name: | Calcitonin gene-related peptide 1 |
|---|
| Synonyms: | CALC1 | CALCA | CALCA_HUMAN | CGRP | Calcitonin gene-related peptide (CGRP alpha) | Calcitonin gene-related peptide 1 |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 13902.80 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P06881 |
|---|
| Residue: | 128 |
|---|
| Sequence: | MGFQKFSPFLALSILVLLQAGSLHAAPFRSALESSPADPATLSEDEARLLLAALVQDYVQ
MKASELEQEQEREGSRIIAQKRACDTATCVTHRLAGLLSRSGGVVKNNFVPTNVGSKAFG
RRRRDLQA
|
|
|
|---|
| BDBM126180 |
|---|
| n/a |
|---|
| Name | BDBM126180 |
|---|
| Synonyms: | US8778957, 61 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C34H35N5O3 |
|---|
| Mol. Mass. | 561.6734 |
|---|
| SMILES | CC(C)(C)OC(=O)N1CCN(Cc2ccc3cc4C[C@@]5(Cc4cc3n2)C(=O)Nc2ncccc52)CC1c1ccccc1 |r| |
|---|
| Structure | 
|
|---|
Search and Browse
