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TargetCalcitonin gene-related peptide (CGRP alpha)
LigandBDBM126188
Substrate/Competitorn/a
Meas. Tech.Binding Assay
pH7.4±n/a
Temperature298.15±n/a K
Ki 1700±n/a nM
Commentsextracted
Citation Stump CAQuigley AG CGRP receptor antagonists US Patent  US8778957 Publication Date 7/15/2014
More Info.:Get all data from this article,  Assay Method
 
Calcitonin gene-related peptide (CGRP alpha)
Name:Calcitonin gene-related peptide (CGRP alpha)
Synonyms:CGRP | Calcitonin gene-related peptide 1
Type:Enzyme
Mol. Mass.:13902.80
Organism:Homo sapiens (Human)
Description:P06881
Residue:128
Sequence:
MGFQKFSPFLALSILVLLQAGSLHAAPFRSALESSPADPATLSEDEARLLLAALVQNYVQ
MKASELEQEQEREGSRIIAQKRACDTATCVTHRLAGLLSRSGGVVKNNFVPTNVGSKAFG
RRRRDLQA
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  Blast E-value cutoff:
BDBM126188
n/a
NameBDBM126188
Synonyms:US8778957, 184
TypeSmall organic molecule
Emp. Form.C25H32N4O2
Mol. Mass.420.5472
SMILESCC(C)[C@H]1CN(C)CCN1Cc1ccc2cc3CC4(Cc3cc2n1)C(C)C(=O)NC4=O |r|
Structure
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