Reaction Details |
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Target | Cannabinoid receptor 2 |
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Ligand | BDBM135909 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Radioligand Binding Assay |
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pH | 7.4±n/a |
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Temperature | 303.15±n/a K |
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Ki | 0.4±n/a nM |
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Comments | extracted |
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Citation | Carroll, WA; Dart, MJ; Frost, JM; Latshaw, SP; Kolasa, T; Li, T; Peddi, S; Liu, B; Perez-Medrano, A; Patel, M; Wang, X; Nelson, DW Compounds as cannabinoid receptor ligands US Patent US8859596 Publication Date 10/14/2014 |
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More Info.: | Get all data from this article, Assay Method |
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Cannabinoid receptor 2 |
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Name: | Cannabinoid receptor 2 |
Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
Type: | G Protein-Coupled Receptor (GPCR) |
Mol. Mass.: | 39690.94 |
Organism: | Homo sapiens (Human) |
Description: | P34972 |
Residue: | 360 |
Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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BDBM135909 |
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n/a |
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Name | BDBM135909 |
Synonyms: | US8859596, 198 |
Type | Small organic molecule |
Emp. Form. | C25H36F3N5O2 |
Mol. Mass. | 495.5808 |
SMILES | CCCCn1n(C)c(c\c1=N/C(=O)c1cc(ccc1NNC(=O)C(C)(C)C)C(F)(F)F)C(C)(C)C |
Structure |
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