| Reaction Details |
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 | Report a problem with these data |
| Target | 5-hydroxytryptamine receptor 1A |
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| Ligand | BDBM136359 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Inhibition Assay |
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| pH | 7.4±n/a |
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| Ki | 0.34±n/a nM |
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| Comments | extracted |
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| Citation |  Andersson, J; Gyback, H; Johansson, A; Linde, CE; Malmstrom, J; Nordvall, G; Weigelt, T; Terp, G 2-carboxamide-7-piperazinyl-benzofuran derivatives US Patent US8859534 Publication Date 10/14/2014 |
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| More Info.: | Get all data from this article, Assay Method |
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| 5-hydroxytryptamine receptor 1A |
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| Name: | 5-hydroxytryptamine receptor 1A |
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| Synonyms: | 5-hydroxytryptamine receptor 1A (5HT1A) |
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| Type: | Protein |
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| Mol. Mass.: | 46351.20 |
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| Organism: | Cricetulus griseus (Chinese hamster) (Cricetulus barabensis griseus) |
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| Description: | G3I1B6 |
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| Residue: | 422 |
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| Sequence: | MDIFSLGQGNNTTSSQEPFGTGGNVTGISDVTFSYQVITSLLLGTLIFCAVLGNACVVAA
IALERSLQNVANYLIGSLAVTDLMVSVLVLPMAALYQVLNKWTLGQVTCDLFIALDVLCC
TSSILHLCAIALDRYWAITDPIDYVNKRTPRRAAALISLTWLIGFLISIPPMLGWRTPED
RSDPDACTISKDHGYTIYSTFGAFYIPLLLMLVLYGRIFRAARFRIRKTVKKVEKKGAST
SLSTSSAPPPKKSLNGQPGNGDWRRSAENRAVGAPCANGAVRQGDDEATLEVIEVHRVGN
SKDHLPLPSESGATSYAPACLERKNERNAEAKRKMALARERKTVKTLGIIMGTFILCWLP
FFIVALVLPFCESSCHMPALLGAIINWLGYSNSLLNPVIYAYFNKDFQNAFKKIIKCKFC
RR
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| BDBM136359 |
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| n/a |
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| Name | BDBM136359 |
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| Synonyms: | US8859534, 45 |
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| Type | Small organic molecule |
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| Emp. Form. | C24H28N4O3 |
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| Mol. Mass. | 420.5041 |
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| SMILES | COc1cccc(CCN2CCN(CC2)c2cccc3cc(oc23)C(=O)N2CCC2)n1 |
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| Structure | 
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