Reaction Details |
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Target | Regulator of G-protein signaling 4 |
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Ligand | BDBM50384773 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Inhibitory Assay |
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IC50 | 93000±n/a nM |
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Citation | Neubig, R; Blazer, L; Husbands, S; Larsen, S; Traynor, J Small molecule inhibitors of RGS proteins US Patent US8865750 Publication Date 10/21/2014 |
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More Info.: | Get all data from this article, Assay Method |
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Regulator of G-protein signaling 4 |
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Name: | Regulator of G-protein signaling 4 |
Synonyms: | RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4) |
Type: | Enzyme |
Mol. Mass.: | 23263.51 |
Organism: | Homo sapiens (Human) |
Description: | P49798 |
Residue: | 205 |
Sequence: | MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
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BDBM50384773 |
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n/a |
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Name | BDBM50384773 |
Synonyms: | CHEMBL2037371 |
Type | Small organic molecule |
Emp. Form. | C18H15NO2 |
Mol. Mass. | 277.3172 |
SMILES | Cc1ccc(cc1)C1=CC(=O)N(Cc2ccccc2)C1=O |t:8| |
Structure |
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