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TargetRegulator of G-protein signaling 4
LigandBDBM136369
Substrate/Competitorn/a
Meas. Tech.Inhibitory Assay
IC50 32000±n/a nM
Citation Neubig, RBlazer, LHusbands, SLarsen, STraynor, J Small molecule inhibitors of RGS proteins US Patent US8865750 Publication Date 10/21/2014
More Info.:Get all data from this article,  Assay Method
 
Regulator of G-protein signaling 4
Name:Regulator of G-protein signaling 4
Synonyms:RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4)
Type:Enzyme
Mol. Mass.:23263.51
Organism:Homo sapiens (Human)
Description:P49798
Residue:205
Sequence:
MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWA
ESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFIS
VQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNP
SSCGAEKQKGAKSSADCASLVPQCA
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BDBM136369
n/a
NameBDBM136369
Synonyms:US8865750, CCG- 203780
TypeSmall organic molecule
Emp. Form.C11H8BrNO2
Mol. Mass.266.091
SMILESBrC1=CC(=O)N(Cc2ccccc2)C1=O |t:1|
Structure
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