Reaction Details | |||
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Target | 5-hydroxytryptamine receptor 5A | ||
Ligand | BDBM148155 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | Binding Assay | ||
pH | 7.4±n/a | ||
Temperature | 310.15±n/a K | ||
Ki | 0.68±n/a nM | ||
Comments | extracted | ||
Citation | Hamaguchi, W; Kinoyama, I; Koganemaru, Y; Miyazaki, T; Kaneko, O; Sekioka, R; Washio, T Tetrahydroisoquinoline derivative US Patent US8962612 Publication Date 2/24/2015 | ||
More Info.: | Get all data from this article, Assay Method | ||
5-hydroxytryptamine receptor 5A | |||
Name: | 5-hydroxytryptamine receptor 5A | ||
Synonyms: | 5-HT-5 | 5-HT-5A | 5-hydroxytryptamine receptor 5 (5-HT5) | 5-hydroxytryptamine receptor 5A (5-HT5A) | 5HT5A_HUMAN | HTR5A | Serotonin (5-HT) receptor | Serotonin receptor 5A | ||
Type: | Enzyme | ||
Mol. Mass.: | 40266.25 | ||
Organism: | Homo sapiens (Human) | ||
Description: | P47898 | ||
Residue: | 357 | ||
Sequence: |
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BDBM148155 | |||
n/a | |||
Name | BDBM148155 | ||
Synonyms: | US8962612, 26 | ||
Type | Small organic molecule | ||
Emp. Form. | C17H14F4N4O | ||
Mol. Mass. | 366.3129 | ||
SMILES | NC(N)=NC(=O)N1CCc2c(F)ccc(c2C1)-c1c(F)cc(F)cc1F |(6,-1.54,;4.67,-.77,;4.67,.77,;3.33,-1.54,;2,-.77,;2,.77,;.67,-1.54,;.67,-3.08,;-.67,-3.85,;-2,-3.08,;-3.33,-3.85,;-3.33,-5.39,;-4.67,-3.08,;-4.67,-1.54,;-3.33,-.77,;-2,-1.54,;-.67,-.77,;-3.33,.77,;-4.67,1.54,;-6,.77,;-4.67,3.08,;-3.33,3.85,;-3.33,5.39,;-2,3.08,;-2,1.54,;-.67,.77,)| | ||
Structure |