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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | 5-hydroxytryptamine receptor 5A | ||
| Ligand | BDBM148163 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | Binding Assay | ||
| pH | 7.4±n/a | ||
| Temperature | 310.15±n/a K | ||
| Ki | 0.75±n/a nM | ||
| Comments | extracted | ||
| Citation |  Hamaguchi, W; Kinoyama, I; Koganemaru, Y; Miyazaki, T; Kaneko, O; Sekioka, R; Washio, T Tetrahydroisoquinoline derivative US Patent US8962612 Publication Date 2/24/2015 | ||
| More Info.: | Get all data from this article, Assay Method | ||
| 5-hydroxytryptamine receptor 5A | |||
| Name: | 5-hydroxytryptamine receptor 5A | ||
| Synonyms: | 5-HT-5 | 5-HT-5A | 5-hydroxytryptamine receptor 5 (5-HT5) | 5-hydroxytryptamine receptor 5A (5-HT5A) | 5HT5A_HUMAN | HTR5A | Serotonin (5-HT) receptor | Serotonin receptor 5A | ||
| Type: | Enzyme | ||
| Mol. Mass.: | 40266.25 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | P47898 | ||
| Residue: | 357 | ||
| Sequence: |
| ||
| BDBM148163 | |||
| n/a | |||
| Name | BDBM148163 | ||
| Synonyms: | US8962612, 66 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C19H17F3N4O | ||
| Mol. Mass. | 374.3597 | ||
| SMILES | NC(N)=NC(=O)N1Cc2c(ccc(F)c2C2(CC2)C1)-c1c(F)cccc1F |(6,-.77,;4.67,,;4.67,1.54,;3.33,-.77,;2,,;2,1.54,;.67,-.77,;-.67,,;-2,-.77,;-3.33,,;-4.67,-.77,;-4.67,-2.31,;-3.33,-3.08,;-3.33,-4.62,;-2,-2.31,;-.67,-3.08,;-1.44,-4.41,;.1,-4.41,;.67,-2.31,;-3.33,1.54,;-4.67,2.31,;-6,1.54,;-4.67,3.85,;-3.33,4.62,;-2,3.85,;-2,2.31,;-.67,1.54,)| | ||
| Structure | 
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