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TargetLymphokine-activated killer T-cell-originated protein kinase
LigandBDBM149038
Substrate/Competitorn/a
Meas. Tech.Kinase Assay
pH7.4±n/a
Temperature298.15±n/a K
IC50 0.88±n/a nM
Commentsextracted
Citation Nakamura, YMatsuo, YHisada, SAhmed, FHuntley, RSajjadi-Hashemi, ZJenkins, DMKargbo, RBCui, WGauuan, PJWalker, JRDecornez, HGurram, M Tricyclic compounds and PBK inhibitors containing the same US Patent US8962648 Publication Date 2/24/2015
More Info.:Get all data from this article,  Assay Method
 
Lymphokine-activated killer T-cell-originated protein kinase
Name:Lymphokine-activated killer T-cell-originated protein kinase
Synonyms:2.7.12.2 | CT84 | Cancer/testis antigen 84 | MAPKK-like protein kinase | Nori-3 | PBK | PDZ-binding kinase | SPK | Spermatogenesis-related protein kinase | T-LAK cell-originated protein kinase | TOPK | TOPK_HUMAN
Type:n/a
Mol. Mass.:36072.55
Organism:Homo sapiens (Human)
Description:n/a
Residue:322
Sequence:
MEGISNFKTPSKLSEKKKSVLCSTPTINIPASPFMQKLGFGTGVNVYLMKRSPRGLSHSP
WAVKKINPICNDHYRSVYQKRLMDEAKILKSLHHPNIVGYRAFTEANDGSLCLAMEYGGE
KSLNDLIEERYKASQDPFPAAIILKVALNMARGLKYLHQEKKLLHGDIKSSNVVIKGDFE
TIKICDVGVSLPLDENMTVTDPEACYIGTEPWKPKEAVEENGVITDKADIFAFGLTLWEM
MTLSIPHINLSNDDDDEDKTFDESDFDDEAYYAALGTRPPINMEELDESYQKVIELFSVC
TNEDPKDRPSAAHIVEALETDV
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BDBM149038
n/a
NameBDBM149038
Synonyms:US8962648, 272
TypeSmall organic molecule
Emp. Form.C21H20N2O2S
Mol. Mass.364.461
SMILESC[C@@H](N(C)C)c1ccc(cc1)-c1c(O)ccc2[nH]c(=O)c3sccc3c12 |r|
Structure
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