| Reaction Details |
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 | Report a problem with these data |
| Target | Ribosyldihydronicotinamide dehydrogenase [quinone] |
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| Ligand | BDBM50156669 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Inhibition of Steady-State Catalysis Assay |
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| IC50 | 79.4±12 nM |
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| Citation |  Leung, KK; Shilton, BH Quinone reductase 2 is an adventitious target of protein kinase CK2 inhibitors TBBz (TBI) and DMAT. Biochemistry54:47-59 (2015) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Ribosyldihydronicotinamide dehydrogenase [quinone] |
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| Name: | Ribosyldihydronicotinamide dehydrogenase [quinone] |
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| Synonyms: | Metallothionein-3 | NMOR2 | NQO2 | NQO2_HUMAN | NRH dehydrogenase [quinone] 2 | NRH:quinone oxidoreductase 2 | QR2 | Quinone reductase 2 | Quinone reductase 2 (NQO2) | Ribosyldihydronicotinamide dehydrogenase [quinone] |
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| Type: | Protein |
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| Mol. Mass.: | 25917.25 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P16083 |
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| Residue: | 231 |
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| Sequence: | MAGKKVLIVYAHQEPKSFNGSLKNVAVDELSRQGCTVTVSDLYAMNLEPRATDKDITGTL
SNPEVFNYGVETHEAYKQRSLASDITDEQKKVREADLVIFQFPLYWFSVPAILKGWMDRV
LCQGFAFDIPGFYDSGLLQGKLALLSVTTGGTAEMYTKTGVNGDSRYFLWPLQHGTLHFC
GFKVLAPQISFAPEIASEEERKGMVAAWSQRLQTIWKEEPIPCTAHWHFGQ
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| BDBM50156669 |
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| n/a |
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| Name | BDBM50156669 |
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| Synonyms: | 4,5,6,7-TETRABROMO-BENZIMIDAZOLE | 4,5,6,7-tetrabromo-1H-benzimidazole | 4,5,6,7-tetrabromo-1H-benzo[d]imidazole | 4,5,6,7-tetrabromo-1Hbenzimidazole (1) | 4,5,6,7-tetrabromobenzimidazole | CHEMBL373937 |
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| Type | Small organic molecule |
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| Emp. Form. | C7H2Br4N2 |
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| Mol. Mass. | 433.72 |
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| SMILES | Brc1c(Br)c(Br)c2[nH]cnc2c1Br |
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| Structure | 
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