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TargetPeptidyl-prolyl cis-trans isomerase B
LigandBDBM286563
Substrate/Competitorn/a
Meas. Tech.Surface Plasmon Resonance (SPR) Assay
pH7.4±n/a
Kd 0.600±n/a nM
Commentsextracted
Citation Fu, JKarur, SLi, XLu, PMergo, WRivkin, ASweeney, ZKTjandra, MWeiss, AYifru, A Cyclic peptides and use as medicines US Patent US9566312 Publication Date 2/14/2017
More Info.:Get all data from this article,  Assay Method
 
Peptidyl-prolyl cis-trans isomerase B
Name:Peptidyl-prolyl cis-trans isomerase B
Synonyms:CYP-S1 | CYPB | Cyclophilin B | Cyclophilin B (CypB) | PPIB | PPIB_HUMAN | PPIase | Peptidyl-prolyl cis-trans isomerase B | Rotamase | S-cyclophilin | SCYLP
Type:Protein
Mol. Mass.:23751.82
Organism:Homo sapiens (Human)
Description:P23284
Residue:216
Sequence:
MLRLSERNMKVLLAAALIAGSVFFLLLPGPSAADEKKKGPKVTVKVYFDLRIGDEDVGRV
IFGLFGKTVPKTVDNFVALATGEKGFGYKNSKFHRVIKDFMIQGGDFTRGDGTGGKSIYG
ERFPDENFKLKHYGPGWVSMANAGKDTNGSQFFITTVKTAWLDGKHVVFGKVLEGMEVVR
KVESTKTDSRDKPLKDVIIADCGKIEVEKPFAIAKE
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  Blast E-value cutoff:
BDBM286563
n/a
NameBDBM286563
Synonyms:US9566312, Compound 2.8.2
TypeSmall organic molecule
Emp. Form.C69H126N12O15S
Mol. Mass.1395.875
SMILESCC[C@H](NC(=O)C([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](NC(=O)[C@@H](NC)[C@H](C)COCCN1CCS(=O)(=O)CC1)C(C)C)C(=O)N(C)[C@H](C)C(C)=O |r|
Structure
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