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TargetPeptidyl-prolyl cis-trans isomerase A
LigandBDBM286606
Substrate/Competitorn/a
Meas. Tech.Surface Plasmon Resonance (SPR) Assay
pH7.4±n/a
Kd 0.900±n/a nM
Commentsextracted
Citation Fu, JKarur, SLi, XLu, PMergo, WRivkin, ASweeney, ZKTjandra, MWeiss, AYifru, A Cyclic peptides and use as medicines US Patent US9566312 Publication Date 2/14/2017
More Info.:Get all data from this article,  Assay Method
 
Peptidyl-prolyl cis-trans isomerase A
Name:Peptidyl-prolyl cis-trans isomerase A
Synonyms:CYPA | CYPA PPIase | Cyclophilin A | Cyclosporin A-binding protein | PPIA | PPIA_HUMAN | PPIase A | Peptidyl-prolyl cis-trans isomerase A | Rotamase A
Type:Protein
Mol. Mass.:18015.32
Organism:Homo sapiens (Human)
Description:P62937
Residue:165
Sequence:
MVNPTVFFDIAVDGEPLGRVSFELFADKVPKTAENFRALSTGEKGFGYKGSCFHRIIPGF
MCQGGDFTRHNGTGGKSIYGEKFEDENFILKHTGPGILSMANAGPNTNGSQFFICTAKTE
WLDGKHVVFGKVKEGMNIVEAMERFGSRNGKTSKKITIADCGQLE
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  Blast E-value cutoff:
BDBM286606
n/a
NameBDBM286606
Synonyms:US9566312, Compound 2.19.2
TypeSmall organic molecule
Emp. Form.C70H125N13O13
Mol. Mass.1356.8208
SMILESCC[C@@H]1NC(=O)[C@H]([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](NC(=O)[C@H]([C@H](C)CCCN2CCC(CC2)C(N)=O)N(C)C(=O)[C@@H](C)N(C)C1=O)C(C)C |r|
Structure
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