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TargetIsoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)
LigandBDBM154558
Substrate/Competitorn/a
Meas. Tech.AlphaScreen Assay
pH8±0
Temperature844.45±0 K
IC50>1.00e+5±n/a nM
Citation Perfetti, MTBaughman, BMDickson, BMMu, YCui, GMader, PDong, ANorris, JLRothbart, SBStrahl, BDBrown, PJJanzen, WPArrowsmith, CHMer, GMcBride, KMJames, LIFrye, SV Identification of a fragment-like small molecule ligand for the methyl-lysine binding protein, 53BP1. ACS Chem Biol10:1072-81 (2015) [PubMed]  Article
More Info.:Get all data from this article,   Solution Info,  Assay Method
 
Isoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)
Name:Isoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)
Synonyms:H-l(3)mbt | H-l(3)mbt protein | KIAA0681 | L(3)mbt protein homolog | L(3)mbt-like | L3MBT | L3MBTL | L3MBTL1 | LMBL1_HUMAN | Lethal(3)malignant brain tumor-like protein 1 | Lethal(3)malignant brain tumor-like protein 1 (4) | Lethal(3)malignant brain tumor-like protein 1 (L3MBTL1)
Type:Protein
Mol. Mass.:83871.06
Organism:Homo sapiens (Human)
Description:Q9Y468-4
Residue:752
Sequence:
MRRREGHGTDSEMGQGPVRESQSSDPPALQFRISEYKPLNMAGVEQPPSPELRQEGVTEY
EDGGAPAGDGEAGPQQAEDHPQNPPEDPNQDPPEDDSTCQCQACGPHQAAGPDLGSSNDG
CPQLFQERSVIVENSSGSTSASELLKPMKKRKRREYQSPSEEESEPEAMEKQEEGKDPEG
QPTASTPESEEWSSSQPATGEKKECWSWESYLEEQKAITAPVSLFQDSQAVTHNKNGFKL
GMKLEGIDPQHPSMYFILTVAEVCGYRLRLHFDGYSECHDFWVNANSPDIHPAGWFEKTG
HKLQPPKGYKEEEFSWSQYLRSTRAQAAPKHLFVSQSHSPPPLGFQVGMKLEAVDRMNPS
LVCVASVTDVVDSRFLVHFDNWDDTYDYWCDPSSPYIHPVGWCQKQGKPLTPPQDYPDPD
NFCWEKYLEETGASAVPTWAFKVRPPHSFLVNMKLEAVDRRNPALIRVASVEDVEDHRIK
IHFDGWSHGYDFWIDADHPDIHPAGWCSKTGHPLQPPLGPREPSSASPGGCPPLSYRSLP
HTRTSKYSFHHRKCPTPGCDGSGHVTGKFTAHHCLSGCPLAERNQSRLKAELSDSEASAR
KKNLSGFSPRKKPRHHGRIGRPPKYRKIPQEDFQTLTPDVVHQSLFMSALSAHPDRSLSV
CWEQHCKLLPGVAGISASTVAKWTIDEVFGFVQTLTGCEDQARLFKDEMIDGEAFLLLTQ
ADIVKIMSVKLGPALKIYNAILMFKNADDTLK
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BDBM154558
n/a
NameBDBM154558
Synonyms:N-(3-(Tert-butylamino)propyl)benzamide (14)
TypeSmall organic molecule
Emp. Form.C14H22N2O
Mol. Mass.234.3373
SMILESCC(C)(C)NCCCNC(=O)c1ccccc1
Structure
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