Reaction Details |
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Target | Trace amine-associated receptor 1 |
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Ligand | BDBM158299 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Radioligand Binding Assay |
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pH | 7.4±n/a |
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Temperature | 310.15±n/a K |
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Ki | 0.5±n/a nM |
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Comments | extracted |
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Citation | Galley, G; Norcross, R; Pflieger, P Substituted benzamide derivatives US Patent US9029370 Publication Date 5/12/2015 |
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More Info.: | Get all data from this article, Assay Method |
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Trace amine-associated receptor 1 |
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Name: | Trace amine-associated receptor 1 |
Synonyms: | TAAR1_MOUSE | Ta1 | Taar1 | Tar1 | Trace amine receptor 1 (TARR1) | Trace amine-associated receptor 1 (TAAR1) | Trace amine-associated receptor1 | Trar1 |
Type: | Protein |
Mol. Mass.: | 37635.41 |
Organism: | Mus musculus (Mouse) |
Description: | Q923Y8 |
Residue: | 332 |
Sequence: | MHLCHAITNISHRNSDWSREVQASLYSLMSLIILATLVGNLIVIISISHFKQLHTPTNWL
LHSMAIVDFLLGCLIMPCSMVRTVERCWYFGEILCKVHTSTDIMLSSASIFHLAFISIDR
YCAVCDPLRYKAKINISTILVMILVSWSLPAVYAFGMIFLELNLKGVEELYRSQVSDLGG
CSPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRTNVQVGLEGKSQAPQ
SKETKAAKTLGIMVGVFLVCWCPFFLCTVLDPFLGYVIPPSLNDALYWFGYLNSALNPMV
YAFFYPWFRRALKMVLLGKIFQKDSSRSKLFL
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BDBM158299 |
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n/a |
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Name | BDBM158299 |
Synonyms: | US9029370, 93 |
Type | Small organic molecule |
Emp. Form. | C21H19ClF2N4O3 |
Mol. Mass. | 448.85 |
SMILES | FC(F)Oc1ccc(cc1)-n1cc(cn1)C(=O)Nc1ccc([C@@H]2CNCCO2)c(Cl)c1 |r| |
Structure |
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