| Reaction Details |
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 | Report a problem with these data |
| Target | Opioid growth factor receptor-like protein 1 |
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| Ligand | BDBM172444 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Radioligand Binding Assay |
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| pH | 7.4±n/a |
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| Temperature | 298.15±n/a K |
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| Ki | 4.2±0.7 nM |
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| Comments | extracted |
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| Citation |  Yamawaki, K; Yao, J; Yu, J; Zhou, X Substituted benzimidazole-type piperidine compounds and uses thereof US Patent US9090618 Publication Date 7/28/2015 |
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| More Info.: | Get all data from this article, Assay Method |
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| Opioid growth factor receptor-like protein 1 |
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| Name: | Opioid growth factor receptor-like protein 1 |
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| Synonyms: | OGFRL1 | OGRL1_HUMAN | Opioid Receptor-Like Receptor (ORL-1) | Opioid growth factor receptor-like protein 1 (ORL-1) | Opioid growth factor receptor-like protein 1 (ORL1) | Opioid receptor-like (ORL-1) | Opioid receptor-like (ORL1) | Opioid receptor-like protein 1 (OGL1) | Opioid receptor-like receptor (ORL1) |
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| Type: | Protein |
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| Mol. Mass.: | 51247.53 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q5TC84 |
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| Residue: | 451 |
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| Sequence: | MGNLLGGVSFREPTTVEDCDSTWQTDSEPEPEEPGPGGGSEGPGQESEQPAQPPEQAGGR
PGASPAPDEDAEAAGAEQGGDSTEATAKPKRSFYAARDLYKYRHQYPNFKDIRYQNDLSN
LRFYKNKIPFKPDGVYIEEVLSKWKGDYEKLEHNHTYIQWLFPLREQGLNFYAKELTTYE
IEEFKKTKEAIRRFLLAYKMMLEFFGIKLTDKTGNVARAVNWQERFQHLNESQHNYLRIT
RILKSLGELGYESFKSPLVKFILHEALVENTIPNIKQSALEYFVYTIRDRRERRKLLRFA
QKHYTPSENFIWGPPRKEQSEGSKAQKMSSPLASSHNSQTSMHKKAKDSKNSSSAVHLNS
KTAEDKKVAPKEPVEETDRPSPEPSNEAAKPRNTEKDSNAENMNSQPEKTVTTPTEKKES
VSPENNEEGGNDNQDNENPGNTNCHDVVLVQ
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| BDBM172444 |
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| n/a |
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| Name | BDBM172444 |
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| Synonyms: | US9090618, ZA67 | US9598411, Ref. No. ZA67 |
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| Type | Small organic molecule |
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| Emp. Form. | C28H36N4O |
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| Mol. Mass. | 444.6116 |
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| SMILES | Cc1cc(no1)-c1nc2ccccc2n1[C@@H]1C[C@@H]2CCC[C@H](C1)N2[C@@H]1C[C@H]2CCC[C@H](C2)C1 |r,THB:24:23:15.16.22:18.20.19| |
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| Structure | 
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