| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
|---|
| Ligand | BDBM181244 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | CB2 Receptor Binding Protocol |
|---|
| Temperature | 303.15±n/a K |
|---|
| Ki | 1.4±0.02 nM |
|---|
| Comments | extracted |
|---|
| Citation |  Moore, II, BM; Bhattacharjee, H; Mustafa, S Tri-aryl/heteroaromatic cannabinoids and use thereof US Patent US9139546 Publication Date 9/22/2015 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Cannabinoid receptor 2 |
|---|
| Name: | Cannabinoid receptor 2 |
|---|
| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
|---|
| Type: | G Protein-Coupled Receptor (GPCR) |
|---|
| Mol. Mass.: | 39690.94 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P34972 |
|---|
| Residue: | 360 |
|---|
| Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
|
|
|
|---|
| BDBM181244 |
|---|
| n/a |
|---|
| Name | BDBM181244 |
|---|
| Synonyms: | US9139546, 42 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C21H18Cl2O |
|---|
| Mol. Mass. | 357.273 |
|---|
| SMILES | CC(C)(c1ccccc1)c1ccc(c(O)c1)-c1cc(Cl)cc(Cl)c1 |
|---|
| Structure | 
|
|---|
Search and Browse
