| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Adenosine receptor A3 [I248L] |
|---|
| Ligand | BDBM191055 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Radioligand Binding Assay |
|---|
| pH | 7.5±n/a |
|---|
| Temperature | 298.15±n/a K |
|---|
| Ki | 12±1 nM |
|---|
| Comments | extracted |
|---|
| Citation |  Jacobson, KA; Tosh, DK Adenosine receptor agonists, partial agonists, and antagonists US Patent US9181253 Publication Date 11/10/2015 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Adenosine receptor A3 [I248L] |
|---|
| Name: | Adenosine receptor A3 [I248L] |
|---|
| Synonyms: | AA3R_HUMAN | ADORA3 | Adenosine receptor A3 | Adenosine receptor A3 (A3) |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 36197.32 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P0DMS8[I248L] |
|---|
| Residue: | 318 |
|---|
| Sequence: | MPNNSTALSLANVTYITMEIFIGLCAIVGNVLVICVVKLNPSLQTTTFYFIVSLALADIA
VGVLVMPLAIVVSLGITIHFYSCLFMTCLLLIFTHASIMSLLAIAVDRYLRVKLTVRYKR
VTTHRRIWLALGLCWLVSFLVGLTPMFGWNMKLTSEYHRNVTFLSCQFVSVMRMDYMVYF
SFLTWIFIPLVVMCAIYLDIFYIIRNKLSLNLSNSKETGAFYGREFKTAKSLFLVLFLFA
LSWLPLSLINCIIYFNGEVPQLVLYMGILLSHANSMMNPIVYAYKIKKFKETYLLILKAC
VVCHPSDSLDTSIEKNSE
|
|
|
|---|
| BDBM191055 |
|---|
| n/a |
|---|
| Name | BDBM191055 |
|---|
| Synonyms: | US9181253, 117 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C14H18ClN5O2 |
|---|
| Mol. Mass. | 323.778 |
|---|
| SMILES | CC(C)Nc1nc(Cl)nc2n(cnc12)[C@]12C[C@H]1[C@@H](O)[C@@H](O)C2 |r| |
|---|
| Structure | 
|
|---|
Search and Browse
