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TargetTrypsin
LigandBDBM50069104
Substrate/Competitorn/a
Meas. Tech.High-Throughput Screening Assay
IC50 19600±2700 nM
Citation Vasioukhin VIChevillet JR Hepsin inhibitors US Patent  US9182402 Publication Date 11/10/2015
More Info.:Get all data from this article,  Assay Method
 
Trypsin
Name:Trypsin
Synonyms:n/a
Type:PROTEIN
Mol. Mass.:24411.24
Organism:Sus scrofa
Description:ChEMBL_1450738
Residue:231
Sequence:
FPTDDDDKIVGGYTCAANSIPYQVSLNSGSHFCGGSLINSQWVVSAAHCYKSRIQVRLGE
HNIDVLEGNEQFINAAKIITHPNFNGNTLDNDIMLIKLSSPATLNSRVATVSLPRSCAAA
GTECLISGWGNTKSSGSSYPSLLQCLKAPVLSDSSCKSSYPGQITGNMICVGFLEGGKDS
CQGDSGGPVVCNGQLQGIVSWGYGCAQKNKPGVYTKVCNYVNWIQQTIAAN
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  Blast E-value cutoff:
BDBM50069104
n/a
NameBDBM50069104
Synonyms:CHEMBL1449583 | US9182402, 4
TypeSmall organic molecule
Emp. Form.C18H16N2
Mol. Mass.260.333
SMILESCc1cccc(c1)C1Nc2cccc3cccc(N1)c23
Structure
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