| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Prolactin-releasing peptide receptor |
|---|
| Ligand | BDBM195749 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Inhibition Assay |
|---|
| pH | 7.4±n/a |
|---|
| Temperature | 298.15±n/a K |
|---|
| Ki | 5±n/a nM |
|---|
| Comments | extracted |
|---|
| Citation |  Takahashi, A; Suzuki, M; Nakamura, Y; Sakurai, Y Heterocyclic compounds for the treatment of stress-related conditions US Patent US9206173 Publication Date 12/8/2015 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Prolactin-releasing peptide receptor |
|---|
| Name: | Prolactin-releasing peptide receptor |
|---|
| Synonyms: | G-protein coupled receptor 10 (GPR10) | GPR10 | GR3 | PRLHR | PRLHR_HUMAN | Prolactin Releasing Peptide Receptor | Prolactin-releasing peptide receptor |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 41138.32 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P49683 |
|---|
| Residue: | 370 |
|---|
| Sequence: | MASSTTRGPRVSDLFSGLPPAVTTPANQSAEASAGNGSVAGADAPAVTPFQSLQLVHQLK
GLIVLLYSVVVVVGLVGNCLLVLVIARVRRLHNVTNFLIGNLALSDVLMCTACVPLTLAY
AFEPRGWVFGGGLCHLVFFLQPVTVYVSVFTLTTIAVDRYVVLVHPLRRRISLRLSAYAV
LAIWALSAVLALPAAVHTYHVELKPHDVRLCEEFWGSQERQRQLYAWGLLLVTYLLPLLV
ILLSYVRVSVKLRNRVVPGCVTQSQADWDRARRRRTFCLLVVIVVVFAVCWLPLHVFNLL
RDLDPHAIDPYAFGLVQLLCHWLAMSSACYNPFIYAWLHDSFREELRKLLVAWPRKIAPH
GQNMTVSVVI
|
|
|
|---|
| BDBM195749 |
|---|
| n/a |
|---|
| Name | BDBM195749 |
|---|
| Synonyms: | US9206173, 95 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C26H23F4N5O3 |
|---|
| Mol. Mass. | 529.4861 |
|---|
| SMILES | CCOn1c(N[C@H](C)c2ccc(cc2)C(F)(F)F)nc2CCN(Cc2c1=O)C(=O)c1ccc(cc1F)C#N |r| |
|---|
| Structure | 
|
|---|
Search and Browse
