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TargetMacrophage colony-stimulating factor 1 receptor [555-568]
LigandBDBM198882
Substrate/Competitorn/a
Meas. Tech.Fluorescence Polarization Competition Immunoassay
pH7.5±n/a
IC50 1.3±n/a nM
Commentsextracted
Citation Illig, CRBallentine, SKChen, JDesjarlais, RLMeegalla, SKWall, MWilson, K Inhibitors of c-fms kinase US Patent US9221797 Publication Date 12/29/2015
More Info.:Get all data from this article,  Assay Method
 
Macrophage colony-stimulating factor 1 receptor [555-568]
Name:Macrophage colony-stimulating factor 1 receptor [555-568]
Synonyms:CSF1R | CSF1R_HUMAN | FMS | FMS (aa 555-568) peptide | FMS Substrate Peptide (aa 555-568) | Macrophage colony-stimulating factor 1 receptor (CSF1R) or (c-fms)
Type:Peptide
Mol. Mass.:1619.64
Organism:Homo sapiens (Human)
Description:P07333 aa 555-568
Residue:14
Sequence:
SYEGNSYTFIDPTQ
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  Blast E-value cutoff:
BDBM198882
n/a
NameBDBM198882
Synonyms:US9221797, 67
TypeSmall organic molecule
Emp. Form.C23H27N5O2
Mol. Mass.405.4928
SMILESCOCCNCC(=C)c1ccc(NC(=O)c2nc(c[nH]2)C#N)c(c1)C1=CCCCC1 |t:26|
Structure
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