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TargetDual specificity protein phosphatase CDC14A
LigandBDBM199180
Substrate/Competitorn/a
Meas. Tech.PTP pNPP Assay
pH7±n/a
Temperature298.15±n/a K
Ki>1000±0.0 nM
Commentsextracted
Citation Zhang, ZZhang, S Inhibitors of protein tyrosine phosphatases US Patent US9217012 Publication Date 12/22/2015
More Info.:Get all data from this article,  Assay Method
 
Dual specificity protein phosphatase CDC14A
Name:Dual specificity protein phosphatase CDC14A
Synonyms:3.1.3.16 | 3.1.3.48 | CC14A_HUMAN | CDC14 cell division cycle 14 homolog A | CDC14A
Type:n/a
Mol. Mass.:66598.40
Organism:Homo sapiens (Human)
Description:Q9UNH5
Residue:594
Sequence:
MAAESGELIGACEFMKDRLYFATLRNRPKSTVNTHYFSIDEELVYENFYADFGPLNLAMV
YRYCCKLNKKLKSYSLSRKKIVHYTCFDQRKRANAAFLIGAYAVIYLKKTPEEAYRALLS
GSNPPYLPFRDASFGNCTYNLTILDCLQGIRKGLQHGFFDFETFDVDEYEHYERVENGDF
NWIVPGKFLAFSGPHPKSKIENGYPLHAPEAYFPYFKKHNVTAVVRLNKKIYEAKRFTDA
GFEHYDLFFIDGSTPSDNIVRRFLNICENTEGAIAVHCKAGLGRTGTLIACYVMKHYRFT
HAEIIAWIRICRPGSIIGPQQHFLEEKQASLWVQGDIFRSKLKNRPSSEGSINKILSGLD
DMSIGGNLSKTQNMERFGEDNLEDDDVEMKNGITQGDKLRALKSQRQPRTSPSCAFRSDD
TKGHPRAVSQPFRLSSSLQGSAVTLKTSKMALSPSATAKRINRTSLSSGATVRSFSINSR
LASSLGNLNAATDDPENKKTSSSSKAGFTASPFTNLLNGSSQPTTRNYPELNNNQYNRSS
NSNGGNLNSPPGPHSAKTEEHTTILRPSYTGLSSSSARFLSRSIPSLQSEYVHY
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  Blast E-value cutoff:
BDBM199180
n/a
NameBDBM199180
Synonyms:US9217012, 10
TypeSmall organic molecule
Emp. Form.C46H62F2N5O9P
Mol. Mass.897.9831
SMILESCCc1ccc(cc1)C(=O)NCCCCC(NC(=O)C(Cc1ccc(cc1)C(F)(F)P(O)(O)=O)NC(=O)C(Cc1ccccc1)NC(=O)COC1CC(C)CCC1C(C)C)C(N)=O
Structure
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