Reaction Details |
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Target | Tyrosine-protein kinase ABL1 [T315I] |
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Ligand | BDBM50322535 |
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Substrate/Competitor | Abltide |
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Meas. Tech. | ABL1 (T315I) Kinase Activity Assay |
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Temperature | 298.15±n/a K |
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IC50 | 1±0 nM |
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Comments | extracted |
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Citation | Wang, Y; Zhao, L; Zhang, D; Wu, F; Bi, S; Gao, Y; Chen, H; Chen, H; Zhang, C; Nan, Y; Liu, Y Heteroaryl alkyne compound and use thereof US Patent US9255107 Publication Date 2/9/2016 |
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More Info.: | Get all data from this article, Assay Method |
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Tyrosine-protein kinase ABL1 [T315I] |
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Name: | Tyrosine-protein kinase ABL1 [T315I] |
Synonyms: | ABL | ABL Mutant (T315I) | ABL1 | ABL1_HUMAN | Abelson murine leukemia viral oncogene homolog 1 | JTK7 | Proto-oncogene c-Abl | Proto-oncogene tyrosine-protein kinase ABL1 | Tyrosine-protein kinase ABL (T315I) | Tyrosine-protein kinase ABL1 (T315I) | c-ABL | c-abl (T315I) | p150 |
Type: | n/a |
Mol. Mass.: | 122909.35 |
Organism: | Homo sapiens (Human) |
Description: | P00519 (T315I) |
Residue: | 1130 |
Sequence: | MLEICLKLVGCKSKKGLSSSSSCYLEEALQRPVASDFEPQGLSEAARWNSKENLLAGPSE
NDPNLFVALYDFVASGDNTLSITKGEKLRVLGYNHNGEWCEAQTKNGQGWVPSNYITPVN
SLEKHSWYHGPVSRNAAEYLLSSGINGSFLVRESESSPGQRSISLRYEGRVYHYRINTAS
DGKLYVSSESRFNTLAELVHHHSTVADGLITTLHYPAPKRNKPTVYGVSPNYDKWEMERT
DITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQ
LLGVCTREPPFYIIIEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFI
HRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKS
DVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNP
SDRPSFAEIHQAFETMFQESSISDEVEKELGKQGVRGAVSTLLQAPELPTKTRTSRRAAE
HRDTTDVPEMPHSKGQGESDPLDHEPAVSPLLPRKERGPPEGGLNEDERLLPKDKKTNLF
SALIKKKKKTAPTPPKRSSSFREMDGQPERRGAGEEEGRDISNGALAFTPLDTADPAKSP
KPSNGAGVPNGALRESGGSGFRSPHLWKKSSTLTSSRLATGEEEGGGSSSKRFLRSCSAS
CVPHGAKDTEWRSVTLPRDLQSTGRQFDSSTFGGHKSEKPALPRKRAGENRSDQVTRGTV
TPPPRLVKKNEEAADEVFKDIMESSPGSSPPNLTPKPLRRQVTVAPASGLPHKEEAGKGS
ALGTPAAAEPVTPTSKAGSGAPGGTSKGPAEESRVRRHKHSSESPGRDKGKLSRLKPAPP
PPPAASAGKAGGKPSQSPSQEAAGEAVLGAKTKATSLVDAVNSDAAKPSQPGEGLKKPVL
PATPKPQSAKPSGTPISPAPVPSTLPSASSALAGDQPSSTAFIPLISTRVSLRKTRQPPE
RIASGAITKGVVLDSTEALCLAISRNSEQMASHSAVLEAGKNLYTFCVSYVDSIQQMRNK
FAFREAINKLENNLRELQICPATAGSGPAATQDFSKLLSSVKEISDIVQR
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BDBM50322535 |
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Abltide |
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Name: | Abltide |
Synonyms: | n/a |
Type: | Protein |
Mol. Mass.: | 1338.59 |
Organism: | Homo sapiens (Human) |
Description: | Peptide substrate Abltide (EAIYAAPFAKKK), purchased from Millipore Corporation, USA. |
Residue: | 12 |
Sequence: | |