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| Reaction Details | |||
|---|---|---|---|
 | Report a problem with these data | ||
| Target | Catenin beta-1 [138-686] | ||
| Ligand | BDBM32102 | ||
| Substrate/Competitor | n/a | ||
| Meas. Tech. | AlphaScreen Assay | ||
| pH | 7.4±n/a | ||
| Temperature | 298.15±n/a K | ||
| Ki | 3650±680 nM | ||
| Comments | extracted | ||
| Citation |  Ji, H; Yu, B; Zhang, M; Guo, W Substituted 1H-indazol-1-ol analogs as inhibitors of beta catenin/Tcf protein-protein interactions US Patent US9284299 Publication Date 3/15/2016 | ||
| More Info.: | Get all data from this article, Assay Method | ||
| Catenin beta-1 [138-686] | |||
| Name: | Catenin beta-1 [138-686] | ||
| Synonyms: | Beta-catenin | CTNB1_HUMAN | CTNNB | CTNNB1 | ||
| Type: | Protein | ||
| Mol. Mass.: | 60127.24 | ||
| Organism: | Homo sapiens (Human) | ||
| Description: | aa 138-686 | ||
| Residue: | 549 | ||
| Sequence: |
| ||
| BDBM32102 | |||
| n/a | |||
| Name | BDBM32102 | ||
| Synonyms: | 1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7(1H,6H)-dione | 1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione | 1,6-dimethylpyrimido[5,4-e][1,2,4]triazine-5,7-quinone | MLS000087831 | SMR000024051 | US9284299, PKF118-310 | US9738628, Compound PKF118-310 | cid_66541 | ||
| Type | Small organic molecule | ||
| Emp. Form. | C7H7N5O2 | ||
| Mol. Mass. | 193.1628 | ||
| SMILES | Cn1ncnc2c1nc(=O)n(C)c2=O | ||
| Structure | 
| ||