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TargetSerine/threonine-protein kinase Chk1 [2-280]
LigandBDBM225359
Substrate/Competitorn/a
Meas. Tech.33P-Radiometric_Method1
Ki 5.9±n/a nM
Citation D3R, DD Abbott CHK1 Kinase D3R D3R Publication Date 6/30/2015
More Info.:Get all data from this article,  Assay Method
 
Serine/threonine-protein kinase Chk1 [2-280]
Name:Serine/threonine-protein kinase Chk1 [2-280]
Synonyms:CHEK1 | CHK1 | CHK1_HUMAN | CHK1_Kinase
Type:n/a
Mol. Mass.:32109.16
Organism:Homo sapiens (Human)
Description:O14757[2-280]
Residue:279
Sequence:
AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKM
LNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYL
HGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKR
REFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLAL
LHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS
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  Blast E-value cutoff:
BDBM225359
n/a
NameBDBM225359
Synonyms:Chk1_95
TypeSmall Organic Molecule
Emp. Form.C22H16N2O2
Mol. Mass.340.3746
SMILESOc1ccc(cc1)-c1ccc(cc1)-c1[nH]nc-2c1Cc1cc(O)ccc-21
Structure
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