| Reaction Details |
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 | Report a problem with these data |
| Target | Serine/threonine-protein kinase Chk1 [2-280] |
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| Ligand | BDBM91831 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | 33P-Radiometric_Method1 |
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| Ki | 57.9±n/a nM |
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| Citation |  D3R, DD Abbott CHK1 Kinase D3R D3R Publication Date 6/30/2015 |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Serine/threonine-protein kinase Chk1 [2-280] |
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| Name: | Serine/threonine-protein kinase Chk1 [2-280] |
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| Synonyms: | CHEK1 | CHK1 | CHK1_HUMAN | CHK1_Kinase |
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| Type: | n/a |
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| Mol. Mass.: | 32109.16 |
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| Organism: | Homo sapiens (Human) |
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| Description: | O14757[2-280] |
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| Residue: | 279 |
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| Sequence: | AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKM
LNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYL
HGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKR
REFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLAL
LHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS
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| BDBM91831 |
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| n/a |
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| Name | BDBM91831 |
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| Synonyms: | Chk1_105 |
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| Type | n/a |
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| Emp. Form. | C21H23ClN6O5 |
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| Mol. Mass. | 474.898 |
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| SMILES | COc1cc(NC(=O)CCCCCCC(O)=O)c(Cl)cc1NC(=O)Nc1cnc(cn1)C#N |
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| Structure | 
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