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TargetCHK1_Kinase
LigandBDBM225364
Substrate/Competitorn/a
Meas. Tech.33P-Radiometric_Method1
Ki 9.06±n/a nM
Citation D3R DD Abbott CHK1 Kinase D3R  221 Publication Date 6/30/2015
More Info.:Get all data from this article,  Assay Method
 
CHK1_Kinase
Name:CHK1_Kinase
Synonyms:n/a
Type:n/a
Mol. Mass.:32109.16
Organism:Homo sapiens (Human)
Description:n/a
Residue:279
Sequence:
AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKM
LNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYL
HGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKR
REFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLAL
LHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS
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  Blast E-value cutoff:
BDBM225364
n/a
NameBDBM225364
Synonyms:Chk1_109
TypeSmall Organic Molecule
Emp. Form.C24H18N6O5
Mol. Mass.470.4369
SMILESCOc1cc(ccc1[N+]([O-])=O)-c1ccc2c(Nc3ccc(NC(=O)c4cc[nH]n4)cc3NC2=O)c1
Structure
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