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TargetSerine/threonine-protein kinase Chk1 [2-280]
LigandBDBM225370
Substrate/Competitorn/a
Meas. Tech.33P-Radiometric_Method1
Ki 11.5±n/a nM
Citation D3R, DD Abbott CHK1 Kinase D3R D3R Publication Date 6/30/2015
More Info.:Get all data from this article,  Assay Method
 
Serine/threonine-protein kinase Chk1 [2-280]
Name:Serine/threonine-protein kinase Chk1 [2-280]
Synonyms:CHEK1 | CHK1 | CHK1_HUMAN | CHK1_Kinase
Type:n/a
Mol. Mass.:32109.16
Organism:Homo sapiens (Human)
Description:O14757[2-280]
Residue:279
Sequence:
AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKM
LNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYL
HGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKR
REFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLAL
LHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS
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  Blast E-value cutoff:
BDBM225370
n/a
NameBDBM225370
Synonyms:Chk1_123
TypeSmall Organic Molecule
Emp. Form.C19H16N6O2
Mol. Mass.360.3693
SMILESCOc1cc2Cc3c(n[nH]c3-c3ccc(cc3)-c3nn[nH]n3)-c2cc1OC
Structure
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