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TargetTyrosine-protein kinase SYK [355-635]
LigandBDBM225525
Substrate/Competitorn/a
Meas. Tech.SYK assay_HTRF
IC50 1.42±n/a nM
Citation D3R, DD GSK SYK Kinase D3R D3R Publication Date 6/30/2015
More Info.:Get all data from this article,  Assay Method
 
Tyrosine-protein kinase SYK [355-635]
Name:Tyrosine-protein kinase SYK [355-635]
Synonyms:KSYK_HUMAN | SYK | SYK Kinase
Type:n/a
Mol. Mass.:32610.83
Organism:Homo sapiens (Human)
Description:P43405[355-635]
Residue:281
Sequence:
PEEIRPKEVYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEANDPALK
DELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIEL
VHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKW
PVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCP
AGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN
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  Blast E-value cutoff:
BDBM225525
n/a
NameBDBM225525
Synonyms:GTC000231A
TypeSmall Organic Molecule
Emp. Form.C24H25N9O2
Mol. Mass.471.5144
SMILESCC(=O)NCCCCN(c1ccnc(Nc2ccc3[nH]c(=O)[nH]c3c2)n1)c1cccc2[nH]ncc12
Structure
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