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TargetTyrosine-protein kinase SYK [355-635]
LigandBDBM225527
Substrate/Competitorn/a
Meas. Tech.SYK assay_HTRF
IC50 1.61±n/a nM
Citation D3R, DD GSK SYK Kinase D3R D3R Publication Date 6/30/2015
More Info.:Get all data from this article,  Assay Method
 
Tyrosine-protein kinase SYK [355-635]
Name:Tyrosine-protein kinase SYK [355-635]
Synonyms:KSYK_HUMAN | SYK | SYK Kinase
Type:n/a
Mol. Mass.:32610.83
Organism:Homo sapiens (Human)
Description:P43405[355-635]
Residue:281
Sequence:
PEEIRPKEVYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEANDPALK
DELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIEL
VHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKW
PVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCP
AGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN
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  Blast E-value cutoff:
BDBM225527
n/a
NameBDBM225527
Synonyms:GTC000233A
TypeSmall Organic Molecule
Emp. Form.C20H18FN7O2S
Mol. Mass.439.466
SMILESCCN(c1cccc2[nH]ncc12)c1nc(Nc2ccc3CNS(=O)(=O)c3c2)ncc1F
Structure
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