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TargetUrokinase-type plasminogen activator [179-424,C299A,N323Q]
LigandBDBM50147092
Substrate/Competitorn/a
Meas. Tech.Photometric_Method1
Ki 450±n/a nM
Citation D3R, DD Abbott Urokinase D3R D3R Publication Date 6/30/2015
More Info.:Get all data from this article,  Assay Method
 
Urokinase-type plasminogen activator [179-424,C299A,N323Q]
Name:Urokinase-type plasminogen activator [179-424,C299A,N323Q]
Synonyms:PLAU | UROK_HUMAN | Urokinase
Type:n/a
Mol. Mass.:27687.84
Organism:Homo sapiens (Human)
Description:P00749[179-424,C299A,N323Q]
Residue:246
Sequence:
IIGGEFTTIENQPWFAAIYRRHRGGSVTYVCGGSLISPCWVISATHCFIDYPKKEDYIVY
LGRSRLNSNTQGEMKFEVENLILHKDYSADTLAHHNDIALLKIRSKEGRCAQPSRTIQTI
ALPSMYNDPQFGTSCEITGFGKEQSTDYLYPEQLKMTVVKLISHRECQQPHYYGSEVTTK
MLCAADPQWKTDSCQGDSGGPLVCSLQGRMTLTGIVSWGRGCALKDKPGVYTRVSHFLPW
IRSHTK
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BDBM50147092
n/a
NameBDBM50147092
Synonyms:8-Amino-naphthalene-2-carboxamidine | 8-amino-2-naphthimidamide | CHEMBL319264 | uPa_15
TypeSmall organic molecule
Emp. Form.C11H11N3
Mol. Mass.185.2251
SMILESNC(=N)c1ccc2cccc(N)c2c1
Structure
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