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TargetMelanocortin receptor 5
LigandBDBM230656
Substrate/Competitorn/a
Meas. Tech.Radioligand Binding Assay
IC50 4000±n/a nM
Citation Blaskovich, MACassidy, PJ Methods of modulating the activity of the MC5 receptor and treatment of conditions related to this receptor US Patent US9340517 Publication Date 5/17/2016
More Info.:Get all data from this article,  Assay Method
 
Melanocortin receptor 5
Name:Melanocortin receptor 5
Synonyms:MC5R_MOUSE | Mc5r | Melanocortin receptor 5 | Melanocortin receptor 5 (MC5R)
Type:Enzyme
Mol. Mass.:36966.58
Organism:Mus musculus (Mouse)
Description:P41149
Residue:325
Sequence:
MNSSSTLTVLNLTLNASEDGILGSNVKNKSLACEEMGIAVEVFLTLGLVSLLENILVIGA
IVKNKNLHSPMYFFVGSLAVADMLVSMSNAWETVTIYLLNNKHLVIADTFVRHIDNVFDS
MICISVVASMCSLLAIAVDRYITIFYALRYHHIMTARRSGVIIACIWTFCISCGIVFIIY
YESKYVIICLISMFFTMLFFMVSLYIHMFLLARNHVKRIAASPRYNSVRQRTSMKGAITL
TMLLGIFIVCWSPFFLHLILMISCPQNVYCSCFMSYFNMYLILIMCNSVIDPLIYALRSQ
EMRRTFKEIVCCHGFRRPCRLLGGY
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  Blast E-value cutoff:
BDBM230656
n/a
NameBDBM230656
Synonyms:US9340517, 105
TypeSmall organic molecule
Emp. Form.C35H40N6O2
Mol. Mass.576.7311
SMILESNC(=N)NCCC[C@H]1N[C@@H](CNC(=O)c2ccc3ccccc3c2)CCN(CC(c2ccccc2)c2ccccc2)C1=O
Structure
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