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TargetCytosol aminopeptidase [33-68,L62W]
LigandBDBM234294
Substrate/Competitorn/a
Meas. Tech.Kinetic Inhibition Assay
pH8.4±0
Temperature298.15±0 K
Ki 2.26e+4±n/a nM
Citation Pícha, JLiboska, RBude?ínský, MJirácek, JPawelczak, MMucha, A Unusual activity pattern of leucine aminopeptidase inhibitors based on phosphorus containing derivatives of methionine and norleucine. J Enzyme Inhib Med Chem26:155-61 (2011) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Cytosol aminopeptidase [33-68,L62W]
Name:Cytosol aminopeptidase [33-68,L62W]
Synonyms:AMPL_PIG | Cytosol aminopeptidase | LAP3 | Leucine aminopeptidase (LAP)
Type:Enzyme
Mol. Mass.:4015.44
Organism:Sus scrofa (Pig)
Description:P28839[33-68,L62W]
Residue:36
Sequence:
TKGLVLGIYSKEKEDDAPQFTSAGENFDKWVSGKLR
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BDBM234294
n/a
NameBDBM234294
Synonyms:Met-P (1)
TypeSmall organic molecule
Emp. Form.C4H12NO3PS
Mol. Mass.185.182
SMILESCSCCC(N)P(O)(O)=O
Structure
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