Reaction Details |
| Report a problem with these data |
Target | Cytosol aminopeptidase [33-68,L62W] |
---|
Ligand | BDBM234299 |
---|
Substrate/Competitor | n/a |
---|
Meas. Tech. | Kinetic Inhibition Assay |
---|
pH | 8.4±0 |
---|
Temperature | 298.15±0 K |
---|
Ki | 2.19e+5±n/a nM |
---|
Citation | Pícha, J; Liboska, R; Bude?ínský, M; Jirácek, J; Pawelczak, M; Mucha, A Unusual activity pattern of leucine aminopeptidase inhibitors based on phosphorus containing derivatives of methionine and norleucine. J Enzyme Inhib Med Chem26:155-61 (2011) [PubMed] Article |
---|
More Info.: | Get all data from this article, Assay Method |
---|
|
Cytosol aminopeptidase [33-68,L62W] |
---|
Name: | Cytosol aminopeptidase [33-68,L62W] |
Synonyms: | AMPL_PIG | Cytosol aminopeptidase | LAP3 | Leucine aminopeptidase (LAP) |
Type: | Enzyme |
Mol. Mass.: | 4015.44 |
Organism: | Sus scrofa (Pig) |
Description: | P28839[33-68,L62W] |
Residue: | 36 |
Sequence: | TKGLVLGIYSKEKEDDAPQFTSAGENFDKWVSGKLR
|
|
|
BDBM234299 |
---|
n/a |
---|
Name | BDBM234299 |
Synonyms: | Nle-ψ[P(O)(OH)O]-L-AlaOMe (7) |
Type | Small organic molecule |
Emp. Form. | C9H20NO5P |
Mol. Mass. | 253.2326 |
SMILES | CCCCC(N)P(O)(=O)O[C@@H](C)C(=O)OC |r| |
Structure |
|