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TargetL-lactate:NAD+ oxidoreductase A (LDH-A4)
LigandBDBM234443
Substrate/Competitorn/a
Meas. Tech.LDH Activity Assay
pH7.4±n/a
IC50 140000±n/a nM
Commentsextracted
Citation Rodríguez-Páez LChena-Taboada MACabrera-Hernández ACordero-Martínez JWong C Oxamic acid analogues as LDH-C4-specific competitive inhibitors. J Enzyme Inhib Med Chem 26:579-86 (2011) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
L-lactate:NAD+ oxidoreductase A (LDH-A4)
Name:L-lactate:NAD+ oxidoreductase A (LDH-A4)
Synonyms:n/a
Type:Enzyme
Mol. Mass.:36502.66
Organism:Mus musculus (Mouse)
Description:P06151
Residue:332
Sequence:
MATLKDQLIVNLLKEEQAPQNKITVVGVGAVGMACAISILMKDLADELALVDVMEDKLKG
EMMDLQHGSLFLKTPKIVSSKDYCVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFI
IPNIVKYSPHCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGV
HALSCHGWVLGEHGDSSVPVWSGVNVAGVSLKSLNPELGTDADKEQWKEVHKQVVDSAYE
VIKLKGYTSWAIGLSVADLAESIMKNLRRVHPISTMIKGLYGINEDVFLSVPCILGQNGI
SDVVKVTLTPEEEARLKKSADTLWGIQKELQF
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  Blast E-value cutoff:
BDBM234443
n/a
NameBDBM234443
Synonyms:N-Ethyl oxamate
TypeSmall organic molecule
Emp. Form.C4H6NO3
Mol. Mass.116.0959
SMILESCCNC(=O)C([O-])=O
Structure
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